Assignee: A/S Ferrosan

Location: Soborg, DK
No. of patents: 39

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Number	Title	Issue Date
5010077	ଲ-carbolin-3-carboxylic acid derivatives useful for treating anxiety and related disorders A ଲ-carbolin-3-carboxylic acid derivative of the formula ##STR1## wherein: X is oxygen, sulphur or NR10, wherein R10 is hydrogen, C1-6 -alkyl, C1-6 -alkenyl, C3-7 -cycloalkyl or C3-7 ...	04/23/1991
4999354	Imidazoquinoxaline compounds and their preparation and use New imidazoquinoxaline compounds having the general formula ##STR1## wherein R3 is ##STR2## wherein R' is C1-6 -alkyl, C3-7 -cycloalkyl or C1-6 -alkoxymethyl; and --A-- is ##STR3## wherein ...	03/12/1991
4985446	Piperidine compounds and pharmaceutical compositions thereof Novel piperidine compounds having the formula ##STR1## wherein R3 is 3,4-methylenedioxyphenyl, aryl or heteroaryl which are optionally substituted with one or more C1-6 -alkyl, C1-6 -alkoxy, C3-8 -cycloalky...	01/15/1991
4977155	1,2,3-triazolo compounds Heterocyclic dihydroxyquinoxaline compounds having the formula ##STR1## wherein R2 is hydrogen, NO2, NH2, CN, halogen, or SO2 NH2 ; --X--Y--Z-- is selected from --N.dbd.N--N3 --,--NR3	12/11/1990
4970232	Aryloxyphenylpropylamines and their preparation and use Novel aryloxyphenylpropylamines having the formula ##STR1## wherein R1 is C3-7 -cycloalkyl, C3-10 -alkyl, or alkenyl which may be straight, branched or cyclic, unsubstituted or substituted with C1-4 -alkoxy...	11/13/1990
4968682	Imidazoquinoxaline compounds and their preparation and use New imidazoquinoxaline compounds having the general formula ##STR1## wherein ##STR2## wherein R' is C1-6 -alkyl, C3-7 -cycloalkyl or C1-6 -alkoxymethyl; and ##STR3## wherein R5 is hydrogen or...	11/06/1990
4962122	Aryloxyphenylpropylamines and their preparation and use Novel aryloxyphenylpropylamines having the formula ##STR1## wherein R1 is C3-7 -cycloalkyl, C3-10 -alkyl, or alkenyl which may be straight, branched or cyclic, unsubstituted or substituted with C1-4 -alkoxy...	10/09/1990
4948794	Cycloalkyl or benzyl-6-substituted-quinoxalinediones Heterocyclic dihydroxyquinoxaline compounds having the formula ##STR1## wherein R1 is C1-12 -alkyl, which may optionally be substituted by hydroxy, formyl, carboxy, carboxylic esters, amides or amines, C3-8 -cycloalky...	08/14/1990
4912108	Pyridoquinoxaline compounds and their preparation and use as glutamate antagonists Heterocyclic dihydroxyquinoxaline compounds having the formula ##STR1## wherein --A-- together with the two carbon atoms denoted as 1 and 2 is selected from ##STR2## R1, R2 and R3 are independently H, halogen, CN...	03/27/1990
4902686	Tricyclic heterocyclic compounds and their use in treating benzodiazepin receptor-related ailments New heterocyclic compounds having the general formula ##STR1## wherein R3 is ##STR2## CO2 R' or CONR'R", wherein R' and R" independently are C1-6 -alkyl, C3-7 -cycloalkyl or C1-6 -alkoxymet...	02/20/1990
4889855	Heterocyclic compounds and their preparation and use Heterocyclic dihydroxyquinoxaline compounds having the formula ##STR1## wherein --A-- together with the two carbon atoms denoted as 1 and 2 is selected from ##STR2## R1, R2 and R3 are independently H, halogen, CN...	12/26/1989
4886797	Heterocyclic compounds and their preparation and use New heterocyclic derivatives having the general formula: ##STR1## wherein X is ##STR2## or CO2 R' wherein R' is C1-6 -alkyl, C3-7 -cycloalkyl, or C1-3 -alkoxymethyl, and --A-- is --(CH2)	12/12/1989
4880799	Heterocyclic compounds and their preparation and use New heterocyclic derivatives havingy the general formula: ##STR1## wherein ##STR2## wherein R' is C1-6 -alkyl, C3-7 -cycloalkyl, or C1-3 -alkoxymethyl, and --A-- is --(CH2)n --Y--(CH2	11/14/1989
4877799	Method of treating calcium overload in brain cells of mammals Novel piperidine compounds having the formula ##STR1## wherein R3 is 3,4-methylenedioxyphenyl, aryl or heteroaryl which are optionally substituted with one or more C1-6 -alkyl, C1-6 -alkoxy, C3-8 -cycloalky...	10/31/1989
4873244	Tricyclic heterocyclic compounds as psychopharmaceuticals New heterocyclic compounds having the general formula ##STR1## wherein ##STR2## CO2 R' or CONR'R", wherein R' and R" independently are C1-6 -alkyl, C3-7 -cycloalkyl or C1-6 -alkoxymethyl; --A-- is --C(...	10/10/1989
4870073	Heterocyclic compounds and their preparation and use New heterocyclic derivatives having the general formula: ##STR1## wherein X is ##STR2## or CO2 R' wherein R' is C1-6 -alkyl, C3-7 -cycloalkyl, or C1-3 -alkoxymethyl, and A-- is --(CH2)...	09/26/1989
4866065	Imidazothienopyrimidines useful in psychopharmaceutical preparations New heterocyclic compounds having the general formula ##STR1## wherein ##STR2## wherein R' is C1-6 -alkyl, C3-7 -cycloalkyl or C1-6 -alkoxymethyl; R4 is C1-6 -alkyl; --S-- is ##STR3## ...	09/12/1989
4845095	4-phenylpiperidine compounds and their use Piperidine compounds having the formula ##STR1## wherein R1 is hydrogen, (C1-6 -alkoxyaryl)alkyl, diphenylmethozy-C1-6 -alkyl, C1-8 -alkyl, C4-10 -cycloalkylalkyl, phenoxy-C1-8 -alkyl,...	07/04/1989
4837241	Lipophillically-substituted piperidine oxadiazolyl compounds and their use in stimulating cognitive functions New piperidine compounds having the formula ##STR1## wherein at least one of R3, R4, and R5 are ##STR2## and the other independently are H, C1-6 -alkyl, wherein R' is H, C1-8 -alkyl, phenyl,...	06/06/1989
4812458	6,7-disubstituted-2,3-dihydroxyquinoxaline compounds, pharmaceutical compositions thereof, and their use as neuroleptics Heterocyclic dihydroxyquinoxaline compounds having the formula ##STR1## wherein R1 is halogen, CN, CF3, ethynyl, or N3 and R2 is SO2 C1-3 -alkyl, CF3, NO2, ethynyl, or CN. ...	03/14/1989
4804669	Treatment of pain with a piperidine A method for treating pain in human or non-human animals, which comprises administering an effective, non-toxic amount of paroxetine or a pharmaceutically acceptable salt thereof, to a sufferer....	02/14/1989
4795749	Imidazopyrroloquinoxaline compounds New heterocyclic compounds having the general formula ##STR1## wherein X is ##STR2## wherein R' is C1-6 -alkyl, C3-7 -cycloalkyl, phenyl, thienyl, or C1-3 -alkoxymethyl, R6 and R7 independe...	01/03/1989
4780539	3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments New heterocyclic compounds having the general formula ##STR1## wherein X is ##STR2## or CO2 R' wherein R' is C1-6 -alkyl, C3-7 -cycloalkyl, or C3-7 -cycloalkymethyl, R6 and R7 in...	10/25/1988
4774245	Imidazoquinoxaline compounds New heterocyclic compounds having the general formula ##STR1## wherein X is ##STR2## wherein R1 is C1-6 -alkyl, Cphd 3-7-cycloalkyl, phenyl, thienyl, or C1-3 -alkoxymethyl, R6 and R7 indepe...	09/27/1988
4772599	Benzodiazepine derivatives and their preparation and use New benzodiazepine derivatives of the general formula ##STR1## wherein X1 and X2 independently are ##STR2## wherein R1 is C1-3 -alkyl, C3-5 -cycloalkyl, C1-3 -alkoxymethyl, C...	09/20/1988
4772696	Oxadiazolyl imidazobenzodiazepine process New oxadiazolyl imidazobenzodiazepine derivatives having the formula ##STR1## wherein R3 has the formula ##STR2## wherein R" is hydrogen, C1-6 alkyl C1-6 alkoxymethyl or C3-6 -cycloalkyl; R4...	09/20/1988
4771051	3-substituted-4,5-dihydro-5-oxo imidazoquinazolines, their preparation, and their use in treating benzodiazepin receptor-related ailments New heterocyclic compounds having the general formula ##STR1## wherein X is ##STR2## or CO2 R' wherein R' is C1-6 -alkyl, C3-7 -cycloalkyl, or C3-7 -cycloalkylmethyl, R6 and R7 i...	09/13/1988
4745122	Method for treating obesity A method for treating obesity in humans or non-human animals, which method comprises administering an effective, non-toxic amount of paroxetine or a pharmaceutically acceptable salt thereof, to obese humans or animals and compositions for use in such trea...	05/17/1988
4745112	Oxadiazolylimidazobenzodiazepine, compositions, and method III The application discloses novel benzodiazepine agonist compounds, namely, compounds having the formula ##STR1## wherein X is F, CF3, CH3, or CN, pharmaceutical compositions thereof, and a method of ameliorating central nervous s...	05/17/1988
4727153	Oxadiazolyl intermediates New oxadiazolyl imidazobenzodiazepine derivatives having the formula ##STR1## wherein R3 has the formula ##STR2## wherein R" is hydrogen, C1-6 alkyl C1-6 alkoxymethyl or C3-6 -cycloalkyl; R4...	02/23/1988
4670433	Oxadiazolyl imidazobenzodiazepine derivatives pharmaceutical compositions thereof, and method of treating therewith New oxadiazolyl imidazobenzodiazepine derivatives having the formula ##STR1## wherein R3 has the formula ##STR2## wherein R" is hydrogen, C1-6 alkyl C1-6 alkoxymethyl or C3-6 - cycloalkyl; R4	06/02/1987
4622321	Oxadiazolylimidazobenzodiazepine, compositions, and method The application discloses a novel benzodiazepine agonist compound, namely, 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-4H-imida zo [1,5-a][1,4]benzodiazepine, pharmaceutical compositions thereof, and a method of ameliorating central n...	11/11/1986
4622320	Oxadiazolylimidazobenzodiazepine, compositions, and method The application discloses novel benzodiazepine agonist compounds, namely, 3-(5-cyclopropyl-1,2,4-oxadiazol-3-yl)-5,6-dihydro-5-methyl-6-oxo-7-halo-4 H-imidazo [1,5-a][1,4]benzodiazepines, pharmaceutical compositions thereof, and a method of ameliorating ce...	11/11/1986
4593036	(-)-Trans-4-(4-fluorophenyl)-3-[(4-methoxyphenoxy)meth yl]-1-methylpiperidine useful as 5-HT potentiator The compound (-)-trans-4-(4-florophenyl)-3-[(4-methoxyphenoxy)methyl]-1-methylpiperidin e and pharmaceutically-acceptable acid addition salts thereof, pharmaceutical compositions thereof, and their use in potentiating the 5-hydroxytryptamine(5-HT) of ...	06/03/1986
4585777	(-)-Trans-4-(4-fluorophenyl)-3-(4-methoxyphenoxy)methylpiperidine for potentiating 5-HT The compound (-)-trans-4-(4-fluorophenyl)-3-(4-methoxyphenoxy)methylpiperidine and pharmaceutically-acceptable acid addition salts thereof, pharmaceutical compositions thereof, and their use in potentiating the 5-hydroxytryptamine(5-HT) of a subject ...	04/29/1986
4571424	Optical resolution of racemic femoxetine A process for the optical resolution of the enantiomers of trans-3-[(4-methoxyphenoxy)-methyl]-1-methyl-4-phenylpiperidine, which involves reaction with an enantiomer of mandelic acid to form a mixture of diastereomeric compounds, precipitating one of the...	02/18/1986
4507313	Oxadiazolyl-imidazo-[1,4]benzodiazepines and their use in treatment of diseases of the central nervous system New oxadiazolyl-imidazo-[1,4]benzodiazepine derivatives having benzodiazepine receptor activity have the formula ##STR1## R' is hydrogen, chlorine, fluorine or nitro in the 7- or 8-position, R1 is hydrogen or lower alkyl of up to 3 carbon ...	03/26/1985
4442113	Long-term weight reduction of obese patients using femoxetine A method for assisting with appetite and weight control and reduction in obese human patients, which comprises the step of orally or rectally administering an appetite-suppressant compound selected from the group consisting of femoxetine and a pharmaceuti...	04/10/1984
4371536	ଲ-Carbolin-3-carboxylic acid derivatives A ଲ-carbolin-3-carboxylic acid derivative of the formula ##STR1## has valuable pharmacological properties when administered to patients, e.g. humans as a drug, have been shown to possess interesting tranquilizing activity....	02/01/1983

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Assignee: A/S Ferrosan