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Patent No. 5996127

Wearable Device For Feeding and Observing Birds and Other Flying Animals

A device for feeding and observing flying animals comprising a hat, a support mounted on the hat and extending outward from the hat, and a feeder mounted on the support.

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Assignee: Pfizer Inc. (


Location: Not specified.
No. of applications: 581

1                      
Application No.Application TitleIssue Date
20080305161INJECTABLE DEPOT FORMULATIONS AND METHODS FOR PROVIDING SUSTAINED RELEASE OF NANOPARTICLE COMPOSITIONS
Pharmaceutical formulations comprising: a compound selected from the group consisting of ziprasidone, having a maximum average particle size; a carrier; and preferably at least two surface stabilizers are disclosed. The present invention also comprises methods of treati...
12/11/2008
20080300273Method of Treating Abnormal Cell Growth
The present invention relates to the use of (R)-3-[1-(2,6-Dichloro-3-fluoro-phenyl)-ethoxy]-5-(1-piperidin-4-yl-1H-pyrazol-4-yl)-pyridin-2-ylamine, a novel c-Met/HGFR inhibitor, for treating abnormal cell growth in mammals. In particular, the invention provides methods ...
12/04/2008
20080300234PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH
The present invention relates to a compound of the formula 1

    • wherein R1-R
12/04/2008
20080299188CONTROLLED RELEASE DOSAGE FORMS COMBINING IMMEDIATE RELEASE AND SUSTAINTED RELEASE OF LOW-SOLUBILITY DRUG
A controlled release dosage form comprises an immediate release portion and an enteric coated sustained release core....
12/04/2008
20080293801Solid Amorphous Dispersions of An Mtp Inhibitor For Treatment of Obesity
A composition comprises a solid amorphous dispersion comprising (S)—N-{2-[benzyl(methyl)amino]-2-oxo-1-phenylethyl}-methyl-5-[4′-(trifluoromethyl)[1,1′-biphenyl]-2-carboxamido]-1H-indole-2-carboxamide and a polymer....
11/27/2008
20080293769Polymorphs of a C-Met/Hgfr Inhibitor
This invention relates to polymorphs of (R)-3-[1-(2,6-Dichloro-3-fluoro-phenyl)-ethoxy]-5-(1-piperidin-4-yl-1H-pyrazol-4-yl)-pyridin-2-ylamine that are useful in the treatment of abnormal cell growth, such as cancer, in mammals. This invention also relates to compositio...
11/27/2008
20080293646MACROLIDES
The invention relates to compounds of Formula (I):

wherein R1, R2 and X are as defined herein. The invention also relates to pharmaceutical compositions and methods of treating bacterial...

11/27/2008
20080293633Pharmaceutical Formulations, Methods, and Dosing Regimens for the Treatment and Prevention of Acute Coronary Syndromes
The invention provides methods and formulations for treating and preventing acute coronary syndromes. The methods of the instant invention provide safe and effective doses of an Apolipoprotein A-I Milano: phospholipid complex to reduce and stabilize atherosclerotic plaq...
11/27/2008
20080292707Pharmaceutical Compositions of Adsorbates of Amorphous Drug
Pharmaceutical compositions comprise a low-solubility drug adsorbed onto a high surface area substrate to form an adsorbate. The compositions in some embodiments include a concentration-enhancing polymer....
11/27/2008
20080287479INHIBITORS OF SERINE PALMITOYLTRANSFERASE
This invention provides compounds of the formula:

useful in the inhibition or modulation of serine palmitoyl transferase and their use in methods of treatment or amelioration of type 2 diabetes, type 1 diabet...

11/20/2008
20080287521Crystalline Forms Of [R-(R*,R*)-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methyl- Ethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic Acid Calcium Salt (2:1)
Novel crystalline forms of [R-(R*,R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid hemi calcium salt designated Form V, Form VI, Form VII, Form VIII, Form IX, Form X, Form XI, Form XII, Form XIII, F...
11/20/2008
20080280879SUBSTITUTED HETEROCYCLIC DERIVATIVES AND THEIR PHARMACEUTICAL USE AND COMPOSITIONS
Compounds of the general Formula I, wherein X1, X2, X3, X4, X5, X6, X7, R1, R2, R4, R5, R6, R7, R8, R9, R...
11/13/2008
20080280877Azetidines
The invention relates to EP2 antagonist azetidines of formula (I)

wherein Ar, R1, X, and Z are as defined herein, to their use in medicine, particularly in the treatment of endometriosis and/or ute...

11/13/2008
20080280875FUSED PHENYL AMIDO HETEROCYCLIC COMPOUNDS
The present invention relates to a compound of formula (I):

or a pharmaceutically acceptable salt or solvate thereof, wherein:

    11/13/2008
    20080269293PYRAZOLE DERIVATIVES AS ANTI-PLATELET AND ANTI-THROMBOTIC AGENTS
    This invention relates to novel compounds of formula (I)

    or stereoisomers or pharmaceutically acceptable salts thereof wherein Y, R1 through R9, and X1 through X7 a...

    10/30/2008
    20080269111METHOD OF TREATING DYSLIPIDEMIC DISORDER
    The invention provides methods of treating or preventing a condition or disorder associated with dyslipidemia with compositions comprising apolipoprotein-sphingomyelin complexes. The methods of the invention permit reduction, by 4- to 20-fold, of the amount of apolipopr...
    10/30/2008
    20080269211Indazole Derivatives
    This invention relates to compounds of the formula (I):

    or pharmaceutically acceptable salts thereof, wherein: R1, R2, R3, A and m are each as described herein and composition...

    10/30/2008
    20080269246METHOD FOR TREATING PEDIATRIC BIPOLAR DISORDER
    The present invention, in one aspect, relates to a method of using piperazinyl-heterocyclic compounds of the formula I, as defined below, for enhancing cognition in a mammal, including a human, for example a mammal afflicted with psychosis, autism, dementia, or mental r...
    10/30/2008
    20080261995Pharmaceutical Combination of a Pde-5 Inhibitor and a 5-Alpha Reductase Inhibitor
    This invention relates to the combined use of a PDE5 inhibitor and a 5-alpha reductase antagonist in the treatment of lower urinary tract symptoms (LUTS), such as urgency, frequency, nocturia and urge incontinence....
    10/23/2008
    20080262056Oxindole Oxazolidinones as Antibacterial Agents
    The present invention relates to novel oxazolidinones derivatives of oxindoles of formula I or a pharmaceutically acceptable salt thereof wherein: Y1 is CH or CF; R1 is —C1-4alkyl, optionally substituted with a fluoro atom, or R1 ...
    10/23/2008
    20080249031CRYSTALLINE FORMS
    The present invention relates to crystalline forms of (3S)-3-[N—(N′-(2-tert-butylphenyl)oxamyl)alaninyl]amino-5-(2′,3′,5′,6′-tetrafluorophenoxy)-4-oxopentanoic acid (see formula I). The invention further relates to pharmaceutical compositions comprising such...
    10/09/2008
    20080249094COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS
    The present invention relates to compounds of the Formula

    wherein R3, R5, R7, U, X, Y and Z are as defined. Compounds of the Formula I have activity inhibiting production of A...

    10/09/2008
    20080242874Direct Aminolysis
    In some aspects, the present invention provides a method of preparing a compound of the formula (I) comprising reacting a mesylate compound of the formula (II) by direct aminolysis with a reagent comprising ammonia. The reaction is preferably carried out in a solvent, s...
    10/02/2008
    20080234303PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF ABNORMAL CELL GROWTH
    The present invention relates to a compound of the formula 1
    or a pharmaceutically acceptable salt thereof, wherein Ar is a group of formula
    and R1, R2, R13, A, K, M, L1, L2, X, Y1, Y
    09/25/2008
    20080234252Compounds Useful in Therapy
    Compounds of formula (I),

    or a pharmaceutically acceptable salt, solvate, ester or amide thereof, wherein

    • R1 represents [CH
    09/25/2008
    20080227781IMIDAZOLE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS
    The present invention relates to compounds of the Formula I

    wherein R1, R2, R3, R4, R6, R7 and A are as defined. Compounds of the Formula I ha...

    09/18/2008
    20080227974Novel Substituted Azetidinones
    Novel azetidinones and pharmaceutical compositions are described, as are the methods of using such compounds and compositions to treat subjects, including humans, suffering from hyperlipidemia, hypercholesterolemia, hypertriglyceridemia and atherosclerosis....
    09/18/2008
    20080221154HIV-INTEGRASE INHIBITORS, PHARMACEUTICAL COMPOSITIONS, AND METHODS FOR THEIR USE
    Bicyclic hydroxamate compounds represented by the Formula I:

    are described. The bicyclic hydroxamate compounds and compositions containing those compounds may be used to inhibit or modulate an enzyme activity...

    09/11/2008
    20080214607HETEROAROMATIC QUINOLINE COMPOUNDS
    The invention pertains to heteroaromatic compounds that serve as effective phosphodiesterase (PDE) inhibitors. In particular, the invention relates to said compounds which are selective inhibitors of PDE10. The invention also relates to intermediates for preparation of ...
    09/04/2008
    20080213375Drying of Drug-Containing Particles
    A secondary drying process is disclosed for removing residual solvent from drug-containing particles that have been formed by solvent-based processes, the secondary drying process utilizing a combination of vacuum, agitation, and a stripping gas....
    09/04/2008
    20080215249Crystallization and structure determination of beta secretase and/or beta secretase-like proteins
    The x-ray crystal structure of human BACE or BACE-like proteins is useful for solving the structure of other molecules or molecular complexes, and identifying and/or designing potential modifiers of human BACE activity....
    09/04/2008
    20080214651Crystalline forms of [R-(R*, R*)]-2-(4-fluorophenyl)-beta,delta-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid calcium salt (2:1)
    Novel crystalline forms of [R—(R*,R*)]-2-(4-fluorophenyl)-β,δ-dihydroxy-5-(1-methylethyl)-3-phenyl-4-[(phenylamino)carbonyl]-1H-pyrrole-1-heptanoic acid hemi calcium salt designated Form V, Form VI, Form VII, Form VIII, Form IX, Form X, Form XI, Form XII, Form XIII,...
    09/04/2008
    20080207755Alpha 2 Delta Ligands For Fibromyalgia and Other Disorders
    This invention relates to a method of treating certain disorders by administering a compound of the formula 1

    or a pharmaceutically acceptable salt thereof, wherein:

    R1

    08/28/2008
    20080207712THIAZOLE-AMINE COMPOUNDS FOR THE TREATMENT OF NEURODEGENERATIVE DISORDERS
    The present invention relates to compounds of the Formula I

    wherein R1, R3, R4, R5, R6 and R7 are as defined. Compounds of the Formula I have ...

    08/28/2008
    20080207665Alpha-(Aryl-or Heteroaryl-Methyl)-Beta-Piperidinopropanoic Acid Compounds as Orl-1-Receptor Antagonists
    This invention provides the compounds of formula (I): or a pharmaceutically acceptable ester or salt thereof, wherein R1 and R2 independently represent hydrogen or the like; R3 represents aryl or the like; —X—Y— represents —CH
    08/28/2008
    20080206257Combined treatment with keratinocyte growth factor and epidermal growth factor inhibitor
    The present invention relates to compositions and methods for treating the epithelial toxicity caused by administering to a human cancer patient an epidermal growth factor receptor (EGFR) inhibitor. The pharmaceutical composition preferably comprises an EGFR inhibitor a...
    08/28/2008
    20080207689Formamide Derivatives For The Treatment of Diseases
    The invention relates to compounds of formula (1)

    and to processes for the preparation of, intermediates used in the preparation of, compositions containing and the uses of, such derivatives. The compounds ac...

    08/28/2008
    20080200490Alpha-(Aryl-or Heteroaryl-Methyl)-Beta-Piperidino Propanamide Compounds as Orl-1-Receptor Antagonists
    This invention provides the compounds of formula (I), or a pharmaceutically acceptable salt thereof, wherein R1 and R2 independently represent hydrogen or the like; R3 and R4 independently represents hydrogen or the like; R
    08/21/2008
    200802004754-Piperazinothieno[2,3-D] Pyrimidine Compounds As Platelet Aggregation Inhibitors
    Compounds and pharmaceutically acceptable salts of the compounds are disclosed, wherein the compounds have the structure of Formula I: (I) wherein A1, A2, A3, A4, A5, A6, A7, A8, X
    08/21/2008
    20080194841Preparation of Optically Pure Beta-Amino Acids Having Affinity for the Alpha-Delta Protein
    Disclosed are materials and methods for preparing optically active β-amino acids, which bind to the alpha-2-delta subunit of a calcium channel and are useful for treating pain, fibromyalgia, and a variety of psychiatric and sleep disorders. The method includes reacting...
    08/14/2008
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